SCHEMBL29629424

SCHEMBL29629424

Cc1c(C(N)=O)cccc1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 1/20 0.53
CTSS P25774 3/20 0.50
PARP1 P09874 4/20 0.46
DHODH Q02127 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
LMNA P02545 1/20 0.44
GAA P10253 1/20 0.44
CD38 P28907 4/20 0.44
CYP3A4 P08684 2/20 0.44
CTSK P43235 1/20 0.43
KCNH2 Q12809 1/20 0.43
PTGS1 P23219 1/20 0.41
AURKA O14965 1/20 0.40
RPS6KB1 P23443 1/20 0.40
AURKB Q96GD4 1/20 0.40
SCN9A Q15858 1/20 0.40
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
PDK2 Q15119 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2576656 1.00 TAS2R14 (0.53) TAS2R14CTSSPARP1DHODHHDAC6
SCHEMBL5490483 0.85 TAS2R14 (0.50) TAS2R14CTSSPARP1DHODHHDAC6
SCHEMBL6173688 0.85 PARP1 (0.53) TAS2R14PARP1LMNAGAACD38
SCHEMBL28052031 0.85 TAS2R14 (0.55) TAS2R14CTSSDHODHHDAC6LMNA
SCHEMBL28192127 0.84 TAS2R14 (0.41) TAS2R14CTSSPARP1DHODHHDAC6
SCHEMBL7348566 0.83 CA2 (0.43) PARP1GAAKDM4EALDH1A1MAPT
SCHEMBL5182718 0.83 TAS2R14 (0.40) TAS2R14CTSSPARP1DHODHHDAC6
SCHEMBL697951 0.83 TAS2R14 (0.67) TAS2R14CTSSDHODHHDAC6LMNA
SCHEMBL12327907 0.83 TAS2R14 (0.54) TAS2R14CTSSDHODHHDAC6LMNA
SCHEMBL29656425 0.83 TAS2R14 (0.54) TAS2R14CTSSDHODHHDAC6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3994138-A1 ESTROGEN-RELATED RECEPTOR ALPHA (ERRalpha) MODULATORS Lead Pharma Holding B.V. (NL) 2022-05-11 EP disclosed