SCHEMBL29630883

SCHEMBL29630883

N#Cc1ccc(C=O)cc1F

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.52
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP11B2 P19099 13/20 0.41
CYP11B1 P15538 12/20 0.41
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL923510 1.00 TRPV4 (0.52) TRPV4ALDH1A1SMN1; SMN2CYP11B2CYP11B1
SCHEMBL7562408 0.86 CYP11B2 (0.47) TRPV4ALDH1A1SMN1; SMN2CYP11B2CYP11B1
SCHEMBL6061330 0.85 KIF11 (0.54) TRPV4CYP11B2CYP11B1
SCHEMBL48778 0.84 PTP4A3 (0.49) TRPV4ALDH1A1SMN1; SMN2EGFR
SCHEMBL10613739 0.83 TRPV4 (0.55) TRPV4CYP11B2CYP11B1
SCHEMBL10613747 0.83 TRPV4 (0.55) TRPV4CYP11B2CYP11B1
SCHEMBL14661910 0.83 AR (0.50) TRPV4
SCHEMBL21676228 0.82 TRPV4 (0.46) TRPV4ALDH1A1CYP11B2CYP11B1
SCHEMBL28606434 0.82 TRPV4 (0.53) TRPV4CYP11B2CYP11B1
SCHEMBL4809997 0.81 SLC22A12 (0.47) TRPV4ALDH1A1SMN1; SMN2CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114507227-A Benzisothiazole compound, preparation method thereof, pharmaceutical composition and application 中国医学科学院药物研究所 2022-05-17 CN disclosed