SCHEMBL29636952

SCHEMBL29636952

COc1c(C)ncnc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.46
MAP4K4 O95819 3/20 0.35
LIMK1 P53667 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PI4KB Q9UBF8 2/20 0.34
KDR P35968 2/20 0.34
PIK3CD O00329 1/20 0.34
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
HCK P08631 1/20 0.34
SRC P12931 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
MTOR P42345 1/20 0.34
PIK3CG P48736 1/20 0.34
EPHB4 P54760 1/20 0.34
PRKDC P78527 1/20 0.34
DHFR P00374 2/20 0.33
PI4KA P42356 1/20 0.33
PI4K2B Q8TCG2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16712814 1.00 PDE5A (0.46) PDE5AMAP4K4LIMK1L3MBTL1PI4KB
SCHEMBL13058679 0.83 CYP1A1 (0.39) PDE5AEGFRSRCMAOA
SCHEMBL6233405 0.77 PDE5A (0.46) PDE5AMAP4K4PI4KBKDRPIK3CD
SCHEMBL1872205 0.76 PDE5A (0.49) PDE5AMAP4K4L3MBTL1PI4KBKDR
SCHEMBL14326156 0.74 PDPK1 (0.39) PDE5AMAOA
SCHEMBL12348218 0.73 TDP1 (0.34) PDE5AMAOA
SCHEMBL12261633 0.73 ALDH1A1 (0.39) PDE5AEGFRMAOA
SCHEMBL16712816 0.73 MAOA (0.33) PDE5AMAOA
SCHEMBL29207868 0.73 MAOA (0.33) PDE5AMAOA
SCHEMBL18312184 0.71 PDE5A (0.41) PDE5API4KBKDRPIK3CDABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022094172-A2 INHIBITORS OF BTK NEWAVE PHARMACEUTICAL INC. (US) 2022-05-05 WO disclosed