SCHEMBL29637645

SCHEMBL29637645

CN1c2ccccc2C(=O)C12CCN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.45
CCR5 P51681 2/20 0.44
TSHR P16473 2/20 0.43
SMARCA2 P51531 1/20 0.43
SMARCA4 P51532 1/20 0.43
PBRM1 Q86U86 1/20 0.43
ALOX15 P16050 1/20 0.43
ATM Q13315 1/20 0.43
GPR119 Q8TDV5 1/20 0.43
PDK2 Q15119 1/20 0.42
CYP11B2 P19099 1/20 0.42
MAPK1 P28482 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PRKCG P05129 1/20 0.42
PRKCB P05771 1/20 0.42
PRKCA P17252 1/20 0.42
PRKCH P24723 1/20 0.42
PRKCE Q02156 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23024326 1.00 BACE1 (0.45) BACE1CCR5TSHRSMARCA2SMARCA4
SCHEMBL21383689 0.82 NOTUM (0.39) MAPK1
SCHEMBL4360931 0.81 HRH3 (0.53) CCR5TSHRALOX15ATMGPR119
SCHEMBL4360934 0.81 HRH3 (0.53) CCR5TSHRALOX15ATMGPR119
SCHEMBL30486636 0.80 CCR5 (0.37) BACE1CCR5TSHRSMARCA2SMARCA4
SCHEMBL23046107 0.80 CCR5 (0.37) BACE1CCR5TSHRSMARCA2SMARCA4
SCHEMBL20511867 0.79 OPRD1 (0.49) TSHRSMARCA2SMARCA4PBRM1ALOX15
SCHEMBL29993143 0.79 OPRD1 (0.49) TSHRSMARCA2SMARCA4PBRM1ALOX15
SCHEMBL26251994 0.77 SIGMAR1 (0.50) TSHRMAPK1
SCHEMBL11536144 0.77 ALDH1A1 (0.47) BACE1TSHRALOX15MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478585-A Nitrogen-containing fused heterocyclic compound and preparation method and application thereof 上海青煜医药科技有限公司 2022-05-13 CN disclosed