SCHEMBL29638516

SCHEMBL29638516

Cc1ccc2c(=O)nc[nH]c2c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.54
CHEK1 O14757 1/20 0.54
PIM1 P11309 1/20 0.54
RPS6KA3 P51812 1/20 0.54
NR4A2 P43354 1/20 0.41
RXFP1 Q9HBX9 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
IDO1 P14902 1/20 0.40
HTR2A P28223 1/20 0.40
KIF11 P52732 1/20 0.39
HTT P42858 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.37
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13003705 1.00 PARP1 (0.54) PARP1CHEK1PIM1RPS6KA3NR4A2
SCHEMBL1507612 0.85 PARP1 (0.54) PARP1CHEK1PIM1RPS6KA3NR4A2
SCHEMBL12489082 0.79 PIM1 (0.51) CHEK1PIM1RPS6KA3SMN1; SMN2IDO1
SCHEMBL2191216 0.78 ALDH1A1 (0.55) PARP1PIM1NR4A2RXFP1SMN1; SMN2
SCHEMBL29798728 0.78 PARP1 (0.50) PARP1CHEK1IDO1HTR2A
SCHEMBL1663769 0.78 PRKCI (0.56) PARP1CHEK1PIM1RPS6KA3SMN1; SMN2
SCHEMBL1663176 0.78 LMNA (0.51) PARP1SMN1; SMN2HTR2AHTTMEN1
SCHEMBL144025 0.78 PARP1 (0.50) PARP1CHEK1PIM1RPS6KA3SMN1; SMN2
SCHEMBL1345856 0.78 PARP1 (0.50) PARP1CHEK1IDO1HTR2A
SCHEMBL28572232 0.77 MMP12 (0.60) RXFP1SMN1; SMN2HTR2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116096718-A Aryl amide compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-05-09 CN disclosed
WO-2022089219-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2022-05-05 WO disclosed