SCHEMBL29638622

SCHEMBL29638622

NC(=O)c1cc(F)cc2cncnc12

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.44
RPS6KB1 P23443 10/20 0.42
AKT1 P31749 4/20 0.42
AURKA O14965 1/20 0.38
AURKB Q96GD4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29638494 0.82 PARP1 (0.51) PARP1RPS6KB1AKT1AURKA
SCHEMBL15544783 0.79 PARP1 (0.41) PARP1RPS6KB1AKT1
SCHEMBL29638640 0.78 PARP1 (0.46) PARP1RPS6KB1AURKA
SCHEMBL27830076 0.77 ALDH1A1 (0.47) PARP1RPS6KB1AURKA
SCHEMBL528715 0.75 PARP1 (0.62) PARP1RPS6KB1AKT1AURKAAURKB
SCHEMBL29558330 0.75 PARP1 (0.62) PARP1RPS6KB1AKT1AURKAAURKB
Hydrochloric Acid SCHEMBL31382875 0.73 PARP1 (0.60) PARP1RPS6KB1AKT1AURKAAURKB
SCHEMBL3265420 0.73 RPS6KB1 (0.43) RPS6KB1AKT1
SCHEMBL20515247 0.73 PARP1 (0.65) PARP1RPS6KB1AURKB
SCHEMBL29936937 0.72 RAB9A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022089219-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2022-05-05 WO disclosed