SCHEMBL29638640

SCHEMBL29638640

COc1cc(C(N)=O)c2ncncc2c1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.46
EGFR P00533 2/20 0.45
RPS6KB1 P23443 10/20 0.45
AURKA O14965 8/20 0.45
KDM4E B2RXH2 2/20 0.43
NNMT P40261 1/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
HPGDS O60760 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29638494 0.80 PARP1 (0.51) PARP1RPS6KB1AURKANNMT
SCHEMBL29638622 0.78 PARP1 (0.44) PARP1RPS6KB1AURKA
SCHEMBL27789401 0.78 PARP1 (0.48) PARP1EGFRRPS6KB1AURKAKDM4E
SCHEMBL29923698 0.77 PARP1 (0.58) PARP1EGFRKDM4E
SCHEMBL20515224 0.77 PARP1 (0.58) PARP1EGFRKDM4E
SCHEMBL1325275 0.76 EGFR (0.51) EGFRCYP11B1CYP11B2
SCHEMBL15544783 0.74 PARP1 (0.41) PARP1RPS6KB1
SCHEMBL30509874 0.73 NNMT (0.45) PARP1RPS6KB1KDM4ENNMT
SCHEMBL31582882 0.73 NNMT (0.45) PARP1RPS6KB1KDM4ENNMT
SCHEMBL27830076 0.72 ALDH1A1 (0.47) PARP1RPS6KB1AURKAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022089219-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2022-05-05 WO disclosed