SCHEMBL29640879

SCHEMBL29640879

CCC(C(=O)O)c1cnc(C)nc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 12/20 0.42
AKR1C2 P52895 12/20 0.42
AKR1C1 Q04828 2/20 0.41
PTGS1 P23219 1/20 0.41
P4HTM Q9NXG6 1/20 0.37
GAA P10253 1/20 0.37
THRB P10828 1/20 0.37
AKR1B10 O60218 1/20 0.35
AKR1C4 P17516 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA1A P35348 1/20 0.35
P2RX7 Q99572 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2434546 0.83 EPHX1 (0.33) GAATHRBALDH1A1KDM4ELMNA
SCHEMBL29640874 0.80 ESR2 (0.38) GAATHRBKDM4ELMNA
SCHEMBL9785383 0.80 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C1PTGS1P4HTM
SCHEMBL9785388 0.80 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C1PTGS1P4HTM
SCHEMBL5296036 0.80 GPR84 (0.43) LMNA
SCHEMBL5296026 0.80 GPR84 (0.43) LMNA
SCHEMBL350463 0.75 AKR1C3 (0.61) AKR1C3AKR1C2AKR1C1PTGS1P4HTM
SCHEMBL1574429 0.74 AKR1C3 (0.58) AKR1C3AKR1C2AKR1C1PTGS1GAA
SCHEMBL510548 0.72 ALDH1A1 (0.56) AKR1C3AKR1C2AKR1C1PTGS1GAA
SCHEMBL564831 0.72 AKR1C3 (0.58) AKR1C3AKR1C2AKR1C1PTGS1AKR1B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218857-B P300/CBP HAT inhibitors and methods of use thereof 星座制药公司 2023-11-21 CN disclosed
CN-114450005-A Compounds for the treatment of neurological disorders 星座制药公司 2022-05-06 CN disclosed