SCHEMBL29640917

SCHEMBL29640917

FC(F)(F)c1ccc2c(c1)CN(c1ccnc(-c3ccncn3)n1)C2

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 1/20 0.39
EIF2AK4 Q9P2K8 10/20 0.37
NAMPT P43490 3/20 0.36
CYP1A2 P05177 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
BACE1 P56817 1/20 0.34
ADRB1 P08588 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640835 0.85 ADORA2A (0.38) TRPV3NAMPTCYP1A2ALDH1A1CYP3A4
SCHEMBL29640818 0.82 ROCK1 (0.35) CYP1A2KDM4EALDH1A1CYP3A4CYP2D6
SCHEMBL29640772 0.81 CYP1A2 (0.39) NAMPTCYP1A2KDM4EALDH1A1CYP3A4
SCHEMBL29640770 0.80 ROCK2 (0.47) CYP1A2ALDH1A1CYP3A4CYP2D6CYP2C19
SCHEMBL29627931 0.69 TRPV1 (0.39) TRPV3NAMPTCYP1A2KDM4EALDH1A1
SCHEMBL28242133 0.62 MPL (0.54)
SCHEMBL4659183 0.62 KIF11 (0.61) CYP2D6
SCHEMBL28174574 0.61 MPL (0.42) CYP3A4CYP2C9
SCHEMBL14937596 0.61 ALDH1A1 (0.40) TRPV3NAMPTCYP1A2ALDH1A1
SCHEMBL27415783 0.61 KMO (0.55) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed