SCHEMBL29640920

SCHEMBL29640920

Fc1cc(C#Cn2ncc3ccccc32)cc(-c2ccnc(N3Cc4ccc(Cl)cc4C3)n2)c1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.36
DPP4 P27487 1/20 0.34
FAAH O00519 1/20 0.34
HCRTR1 O43613 2/20 0.33
HCRTR2 O43614 2/20 0.33
ROCK1 Q13464 1/20 0.31
DKK1 O94907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640781 0.92 ROCK2 (0.37) ROCK2FAAHHCRTR1HCRTR2ROCK1
SCHEMBL29640968 0.90 FAAH (0.34) ROCK2FAAHROCK1DKK1
SCHEMBL29640782 0.88 ROCK2 (0.41) ROCK2FAAHHCRTR1HCRTR2ROCK1
SCHEMBL29640788 0.86 ALDH1A1 (0.38) FAAH
SCHEMBL29627711 0.77 ROCK2 (0.55) ROCK2ROCK1
SCHEMBL29640793 0.77 ROCK2 (0.38) ROCK2FAAHHCRTR1HCRTR2ROCK1
SCHEMBL29640778 0.76 ROCK2 (0.38) ROCK2HCRTR1HCRTR2ROCK1
SCHEMBL29640810 0.71 DYRK1A (0.36) ROCK2
SCHEMBL29640858 0.71 DYRK1A (0.33)
SCHEMBL29640878 0.71 DYRK1A (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed