SCHEMBL29646334

SCHEMBL29646334

NNC(=O)c1cccnc1C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.58
HDAC6 Q9UBN7 1/20 0.58
ALDH1A1 P00352 2/20 0.50
KDM4E B2RXH2 1/20 0.43
CD38 P28907 1/20 0.42
ACKR3 P25106 3/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
CTSD P07339 1/20 0.40
KDR P35968 1/20 0.40
NAPRT Q6XQN6 2/20 0.40
PRKCI P41743 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1447540 1.00 P2RX7 (0.58) P2RX7HDAC6ALDH1A1KDM4ECD38
SCHEMBL7988780 0.83 HDAC6 (0.58) P2RX7HDAC6ALDH1A1KDM4ECD38
SCHEMBL4372942 0.83 HDAC6 (0.51) P2RX7HDAC6ALDH1A1KDM4ECD38
SCHEMBL2148942 0.81 HDAC6 (0.48) P2RX7HDAC6ALDH1A1KDM4ECD38
SCHEMBL30477668 0.81 HDAC6 (0.48) P2RX7HDAC6ALDH1A1KDM4ECD38
SCHEMBL628397 0.81 PARP1 (0.51) HDAC6ALDH1A1KDM4ECD38HTT
SCHEMBL29687007 0.81 PARP1 (0.51) HDAC6ALDH1A1KDM4ECD38HTT
SCHEMBL27764496 0.80 HDAC6 (0.50) HDAC6ALDH1A1KDM4ECD38HTT
SCHEMBL4394779 0.80 HDAC6 (0.51) HDAC6ALDH1A1HCRTR1HCRTR2
Hydrochloric Acid SCHEMBL6828318 0.79 PARP1 (0.50) HDAC6ALDH1A1KDM4ECD38HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN disclosed