SCHEMBL29646374

SCHEMBL29646374

COc1ccccc1-c1nc2c3ccccc3nc(Cl)n2n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 0.49
CYP3A4 P08684 9/20 0.49
CYP2D6 P10635 8/20 0.49
TSHR P16473 6/20 0.49
HSD17B10 Q99714 6/20 0.49
USP2 O75604 6/20 0.49
LMNA P02545 5/20 0.49
ALDH1A1 P00352 5/20 0.49
MAPK1 P28482 4/20 0.49
CYP2C19 P33261 4/20 0.49
ALOX15 P16050 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
TP53 P04637 2/20 0.49
KDM4E B2RXH2 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
CLK4 Q9HAZ1 3/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ADORA2A P29274 1/20 0.45
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25118631 1.00 CYP1A2 (0.49) CYP1A2CYP3A4CYP2D6TSHRHSD17B10
SCHEMBL22987934 0.86 ADORA3 (0.51) TSHRALDH1A1KDM4EMEN1KMT2A
SCHEMBL22979556 0.85 ADORA3 (0.40) HSD17B10LMNAALDH1A1SMN1; SMN2TP53
SCHEMBL29646313 0.85 ADORA3 (0.40) HSD17B10LMNAALDH1A1SMN1; SMN2TP53
SCHEMBL29646400 0.85 C1R (0.42) ADORA3ADORA1MAPTC1R
SCHEMBL22987859 0.85 ADORA3 (0.42) ALDH1A1SMN1; SMN2TP53MEN1KMT2A
SCHEMBL22979544 0.85 C1R (0.42) ADORA3ADORA1MAPTC1R
SCHEMBL22980067 0.83 TP53 (0.47) MAPK1TP53ADORA2APOLBADORA3
SCHEMBL22979102 0.83 ADORA3 (0.50) CYP1A2CYP3A4CYP2D6TSHRHSD17B10
SCHEMBL29646419 0.83 TP53 (0.47) MAPK1TP53ADORA2APOLBADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114466850-B [1,2,4] Triazolo [1,5-C ] quinazolin-5-amine 拜耳股份有限公司 2024-09-10 CN disclosed
CN-114466850-A [1,2,4] triazolo [1,5-C ] quinazolin-5-amines 拜耳股份有限公司 2022-05-10 CN disclosed