SCHEMBL29648992

SCHEMBL29648992

COC(=O)c1ccc(OC)cc1C(F)(F)F.COc1ccc(C(=O)NN)c(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 7/20 0.50
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CFTR P13569 2/20 0.46
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
ESRRA P11474 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TP53 P04637 1/20 0.42
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42
TUBA4A P68366 1/20 0.42
TUBB4B P68371 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2633928 0.94 EPHX2 (0.54) EPHX2KDM4EALDH1A1POLBSMN1; SMN2
SCHEMBL22979384 0.90 KDM4E (0.51) EPHX2KDM4EALDH1A1CFTRCA1
SCHEMBL13784795 0.78 THRB (0.59) ALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL4841210 0.78 THRA (0.47) EPHX2CFTRESRRACYP1A2CYP2C9
SCHEMBL30938349 0.78 KDM4E (0.59) EPHX2KDM4ESMN1; SMN2CFTRCA1
SCHEMBL5460005 0.78 MAPK10 (0.53) EPHX2KDM4EALDH1A1CA1CA2
SCHEMBL5729973 0.78 EPHX2 (0.48) EPHX2ALDH1A1SMN1; SMN2MAPK10P2RX1
SCHEMBL8346226 0.78 KDM4E (0.51) KDM4EALDH1A1SMN1; SMN2CFTRCA1
SCHEMBL14157044 0.78 RAB9A (0.57) EPHX2KDM4EALDH1A1SMN1; SMN2CA1
SCHEMBL1983309 0.78 AKR1C3 (0.53) EPHX2KDM4EALDH1A1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4013508-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES Bayer Aktiengesellschaft (DE) 2022-06-22 EP disclosed