SCHEMBL29654075

SCHEMBL29654075

COc1cccc(-c2csc(-c3csc(N)n3)n2)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.67
CYP1A1 P04798 6/20 0.65
CYP1B1 Q16678 6/20 0.65
CYP1A2 P05177 5/20 0.65
LTA4H P09960 1/20 0.60
RAB9A P51151 4/20 0.57
MAPT P10636 4/20 0.57
ALDH1A1 P00352 4/20 0.57
NPC1 O15118 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
POLB P06746 1/20 0.57
ATP4A P20648 1/20 0.57
ATP4B P51164 1/20 0.57
SREBF2 Q12772 1/20 0.57
PLG P00747 1/20 0.55
PLAT P00750 1/20 0.55
PRSS1 P07477 1/20 0.55
C1S P09871 1/20 0.55
HPGD P15428 2/20 0.53
HTT P42858 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL235435 0.93 LTA4H (0.67) CYP19A1CYP1A1CYP1B1CYP1A2LTA4H
SCHEMBL1180783 0.87 CYP19A1 (0.76) CYP19A1CYP1A1CYP1B1CYP1A2RAB9A
SCHEMBL29654031 0.85 CYP1B1 (0.73) CYP19A1CYP1A1CYP1B1CYP1A2LTA4H
SCHEMBL1180576 0.83 CYP19A1 (0.71) CYP19A1CYP1A1CYP1B1CYP1A2RAB9A
SCHEMBL29654110 0.82 MAPT (0.84) CYP19A1CYP1A1CYP1B1LTA4HRAB9A
SCHEMBL1181045 0.80 CYP19A1 (0.67) CYP19A1CYP1A1CYP1B1RAB9AMAPT
SCHEMBL29654017 0.79 ALDH1A1 (0.66) CYP1A1CYP1B1CYP1A2LTA4HRAB9A
SCHEMBL29654020 0.78 CYP19A1 (0.65) CYP19A1CYP1A1CYP1B1CYP1A2LTA4H
SCHEMBL29654203 0.78 KDM4E (0.85) CYP1A1CYP1B1CYP1A2RAB9AMAPT
SCHEMBL22801080 0.78 RAB9A (0.73) LTA4HRAB9AMAPTALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed