SCHEMBL29657643

SCHEMBL29657643

Cc1cccc(-n2cc(-c3ccc(C=O)cc3)nn2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.61
KEAP1 Q14145 2/20 0.58
NFE2L2 Q16236 2/20 0.58
HSD17B1 P14061 1/20 0.52
HSD17B2 P37059 1/20 0.52
CA2 P00918 4/20 0.51
CA1 P00915 3/20 0.51
CA12 O43570 3/20 0.51
CA9 Q16790 3/20 0.51
CA5A P35218 2/20 0.50
CA5B Q9Y2D0 2/20 0.50
FLT3 P36888 2/20 0.50
GSK3B P49841 1/20 0.50
KDM4E B2RXH2 1/20 0.49
KDM6B O15054 1/20 0.49
KDM5C P41229 1/20 0.49
KDM4C Q9H3R0 1/20 0.49
KDM2A Q9Y2K7 1/20 0.49
KDM3A Q9Y4C1 1/20 0.49
PTGS2 P35354 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28408538 1.00 KDR (0.61) KDRKEAP1NFE2L2HSD17B1HSD17B2
SCHEMBL31473225 0.86 KEAP1 (0.62) KDRKEAP1NFE2L2HSD17B1HSD17B2
SCHEMBL28408386 0.85 FLT3 (0.69) KDRKEAP1NFE2L2HSD17B1HSD17B2
SCHEMBL29657637 0.85 FLT3 (0.69) KDRKEAP1NFE2L2HSD17B1HSD17B2
SCHEMBL28418357 0.84 STS (0.62) KDRKEAP1NFE2L2HSD17B1HSD17B2
SCHEMBL29657629 0.84 STS (0.62) KDRKEAP1NFE2L2HSD17B1HSD17B2
SCHEMBL28418132 0.83 PTGS2 (0.64) KDRCA2CA1CA12CA9
SCHEMBL4549459 0.83 P2RX7 (0.58) KDRKEAP1NFE2L2HSD17B1HSD17B2
SCHEMBL23557659 0.82 HSD17B1 (0.76) KDRKEAP1NFE2L2HSD17B1HSD17B2
SCHEMBL31473210 0.82 KDR (0.60) KDRKEAP1NFE2L2HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111153889-B 2-indolone-triazole anti-tumor compound and preparation method and application thereof 中国医科大学 2022-05-20 CN disclosed