SCHEMBL29673142

SCHEMBL29673142

COC(=O)C1CCCc2ccc(Cl)cc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4C Q9H3R0 1/20 0.42
PTGDR Q13258 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TAS1R2 Q8TE23 1/20 0.41
SIRT1 Q96EB6 4/20 0.41
ACHE P22303 1/20 0.40
SIRT2 Q8IXJ6 2/20 0.40
SIRT3 Q9NTG7 2/20 0.40
HTR2A P28223 3/20 0.39
HTR2C P28335 3/20 0.39
HTR2B P41595 3/20 0.39
ADRB1 P08588 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24542973 1.00 LMNA (0.43) LMNAMEN1MAPTKMT2AKDM4C
SCHEMBL19469643 0.91 HTR2B (0.41) PTGDRPTGDR2HTR2AHTR2CHTR2B
SCHEMBL24542982 0.89 KDM4C (0.42) LMNAMEN1MAPTKMT2AKDM4C
SCHEMBL22652430 0.83 KMT2A (0.41) LMNAMEN1MAPTKMT2AACHE
SCHEMBL5847603 0.83 MTNR1A (0.54)
SCHEMBL28766567 0.82 KDM4C (0.46) KDM4CPTGDRPTGDR2TAS1R3TAS1R1
SCHEMBL29673179 0.82 KDM4C (0.46) KDM4CPTGDRPTGDR2TAS1R3TAS1R1
SCHEMBL1061933 0.81 SIRT1 (0.54) MEN1MAPTKMT2AKDM4CTAS1R3
SCHEMBL29552779 0.79 P2RX7 (0.46) HTR2AHTR2CHTR2B
SCHEMBL23670494 0.79 P2RX7 (0.46) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114644631-A KRAS G12C protein mutation inhibitor, preparation method thereof, pharmaceutical composition and application thereof 上海维申医药有限公司 2022-06-21 CN disclosed