SCHEMBL29680865

SCHEMBL29680865

COc1ccc(-n2ccc3c(-c4ccc(CNCCC(C)N(C)C)cc4)nc(-c4ccc(CNCCC(C)N(C)C)cc4)nc32)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.41
ALDH1A1 P00352 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPSR1 Q6W5P4 2/20 0.38
GAA P10253 1/20 0.38
CCNB2 O95067 1/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
CCNB3 Q8WWL7 1/20 0.38
MEN1 O00255 6/20 0.37
KMT2A Q03164 6/20 0.37
MITF O75030 1/20 0.36
LMNA P02545 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
GPR35 Q9HC97 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
XBP1 P17861 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL29680212 0.95 ALDH1A1 (0.39) MAPK1ALDH1A1L3MBTL1NPSR1GAA
SCHEMBL29680662 0.90 HDAC1 (0.33) MAPK1ALDH1A1NPSR1CDK1MEN1
SCHEMBL29680538 0.89 LSS (0.32) MAPK1ALDH1A1NPSR1CDK1MEN1
Oxalic Acid SCHEMBL29680298 0.86 HDAC1 (0.36) MAPK1ALDH1A1GAACDK1MEN1
Oxalic Acid SCHEMBL29680606 0.85 KDM4E (0.36) MAPK1ALDH1A1GAAMEN1KMT2A
SCHEMBL29680879 0.80 TDP2 (0.32) MAPK1ALDH1A1NPSR1GAALMNA
SCHEMBL29680755 0.79 ABL1 (0.33) CDK1MEN1KMT2ALMNAPDE4B
SCHEMBL29680480 0.78 TDP2 (0.32) MAPK1ALDH1A1NPSR1GAAMEN1
SCHEMBL29680517 0.78 LMNA (0.41) MAPK1ALDH1A1LMNANOS2PDE4B
Oxalic Acid SCHEMBL29680389 0.77 KDM4E (0.37) ALDH1A1GAAMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP claimed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO claimed
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed