SCHEMBL2968658

SCHEMBL2968658

CN(C(=O)OCc1ccccc1)[C@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.59
ITGA2B P08514 1/20 0.59
ABCB1 P08183 2/20 0.57
ALDH1A1 P00352 5/20 0.49
CTRB1 P17538 2/20 0.47
P2RX7 Q99572 1/20 0.46
CTSL P07711 2/20 0.46
CTSB P07858 2/20 0.46
CTSS P25774 2/20 0.46
CTSK P43235 2/20 0.46
MAPT P10636 2/20 0.46
HPGD P15428 1/20 0.46
FOLH1 Q04609 1/20 0.46
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31739224 1.00 ITGB3 (0.59) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL2494968 1.00 ITGB3 (0.59) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL8067076 1.00 ITGB3 (0.59) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL26654521 0.98 ITGB3 (0.58) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL26654515 0.98 ITGB3 (0.58) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL30688507 0.94 ITGB3 (0.58) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL30688544 0.94 ITGB3 (0.58) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL30688553 0.94 ITGB3 (0.58) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL25183099 0.93 ITGB3 (0.57) ITGB3ITGA2BABCB1ALDH1A1CTRB1
SCHEMBL25186398 0.92 ITGB3 (0.53) ITGB3ITGA2BABCB1ALDH1A1CTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7767811-B2 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids BRANDEIS UNIVERSITY (US) 2010-08-03 US disclosed
US-20060293536-A1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids BRANDEIS UNIVERSITY (US) 2006-12-28 US disclosed
US-7057038-B2 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids BRANDEIS UNIVERSITY (US) 2006-06-06 US disclosed
EP-1419125-A4 KINETIC RESOLUTIONS OF CHIRAT 3- AND 3-SUBSTITUTED CARBOXYLIC ACIDS UNIV BRANDEIS (US) 2005-03-23 EP disclosed
US-20050020849-A1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids DENG LI (US) 2005-01-27 US disclosed
US-6743914-B2 USING TERTIARY AMINE CATALYST BRANDEIS UNIVERSITY 2004-06-01 US disclosed
EP-1419125-A1 KINETIC RESOLUTIONS OF CHIRAT 3- AND 3-SUBSTITUTED CARBOXYLIC ACIDS Brandeis University (US) 2004-05-19 EP disclosed
EP-1305270-B1 KINETIC RESOLUTIONS OF CHIRAL 2- AND 3-SUBSTITUTED CARBOXYLIC ACIDS UNIV BRANDEIS (US) 2004-04-14 EP disclosed
US-20030166963-A1 Kinetic resolutions of chiral 2-and 3-substituted carboxylic acids NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-09-04 US disclosed
US-6562967-B2 Drug screening; purity BRANDEIS UNIVERSITY 2003-05-13 US disclosed
EP-1305270-A1 KINETIC RESOLUTIONS OF CHIRAL 2- AND 3-SUBSTITUTED CARBOXYLIC ACIDS Brandeis University (US) 2003-05-02 EP disclosed
WO-2003011799-A1 KINETIC RESOLUTIONS OF CHIRAT 3- AND 3-SUBSTITUTED CARBOXYLIC ACIDS BRANDEIS UNIVERSITY (US) 2003-02-13 WO disclosed
US-20020165393-A1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2002-11-07 US disclosed
US-20020151744-A1 Kinetic resolutions of chiral 2-and-3-substituted carboxylic acids NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2002-10-17 US disclosed
WO-2002010096-A1 KINETIC RESOLUTIONS OF CHIRAL 2- AND 3-SUBSTITUTED CARBOXYLIC ACIDS BRANDEIS UNIVERSITY (US) 2002-02-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020165393-A1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids ADH5, ADH1C, TST ITGB3 1780/4885ITGA2B 3170/4885ABCB1 4828/4885
US-20050020849-A1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids ADH5, ADH1C, TST ITGB3 1008/4885ITGA2B 2236/4885ABCB1 4760/4885
US-20060293536-A1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids ADH5, ADH1C, TST ITGB3 1008/4885ITGA2B 2236/4885ABCB1 4760/4885
US-20030166963-A1 Kinetic resolutions of chiral 2-and 3-substituted carboxylic acids ADH5, ADH1C, TST ITGB3 1859/4885ITGA2B 3225/4885ABCB1 4832/4885
US-20020151744-A1 Kinetic resolutions of chiral 2-and-3-substituted carboxylic acids ADH5, ADH1C, TST ITGB3 1272/4885ITGA2B 2689/4885ABCB1 4791/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.