SCHEMBL29689869

SCHEMBL29689869

O=Cc1cc(Br)ccc1OCc1ccc(Cl)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.63
PTGDR2 Q9Y5Y4 1/20 0.55
STAT3 P40763 1/20 0.54
NPSR1 Q6W5P4 1/20 0.53
TACR2 P21452 1/20 0.52
SLC6A4 P31645 1/20 0.52
MEN1 O00255 1/20 0.52
PLA2G1B P04054 1/20 0.52
POLB P06746 1/20 0.52
DNMT1 P26358 1/20 0.52
GFER P55789 1/20 0.52
KMT2A Q03164 1/20 0.52
ATG4B Q9Y4P1 1/20 0.52
NPC1 O15118 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
MAPT P10636 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5699666 1.00 CCR5 (0.63) CCR5PTGDR2STAT3NPSR1TACR2
SCHEMBL29227218 0.91 CCR5 (0.56) CCR5PTGDR2STAT3NPSR1TACR2
SCHEMBL30679658 0.88 CCR5 (0.59) CCR5STAT3NPSR1TACR2SLC6A4
SCHEMBL5699833 0.85 LMNA (0.69) CCR5PTGDR2NPC1ALDH1A1LMNA
SCHEMBL5700125 0.85 PTGDR2 (0.55) CCR5PTGDR2NPC1ALDH1A1LMNA
SCHEMBL30866193 0.85 CCR5 (0.62) CCR5PTGDR2NPSR1MEN1POLB
SCHEMBL275887 0.85 CCR5 (0.62) CCR5PTGDR2NPSR1MEN1POLB
SCHEMBL82269 0.85 PTGDR2 (0.61) CCR5PTGDR2SLC6A4NPC1ALDH1A1
SCHEMBL29690396 0.85 PTGDR2 (0.61) CCR5PTGDR2SLC6A4NPC1ALDH1A1
SCHEMBL2284584 0.85 CCR5 (0.65) CCR5PTGDR2SLC6A4CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114671815-B Aryl barbiturates compound and preparation method and application thereof 中国医学科学院药物研究所 2024-05-14 CN disclosed
CN-117430570-A Rhodamine acetic acid compound, and pharmaceutical composition and application thereof 中国医学科学院药物研究所 2024-01-23 CN disclosed
CN-114671815-A Aryl barbiturates compound and preparation method and application thereof 中国医学科学院药物研究所 2022-06-28 CN disclosed