SCHEMBL29756368

SCHEMBL29756368

Cc1nc(-c2ccc(OCCn3cc(Br)cn3)cc2)cc2c1[nH]c1ccc(Cl)cc12

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.36
ACHE P22303 6/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
CXCR1 P25024 2/20 0.34
TBK1 Q9UHD2 1/20 0.32
MAOA P21397 2/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
DRD3 P35462 1/20 0.31
MCHR1 Q99705 1/20 0.31
PLA2G4A P47712 1/20 0.31
MGAM O43451 1/20 0.31
GAA P10253 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20122753 0.80 TBK1 (0.33) ACHECYP1A2CYP2C19TBK1MAOA
SCHEMBL20122733 0.77 MAOA (0.42) ACHECYP1A2MAOAKDM4EALDH1A1
SCHEMBL29756399 0.70 MEN1 (0.40) CYP1A2CYP2C19KDM4EALDH1A1GAA
SCHEMBL23097174 0.67 PRKAB2 (0.31)
SCHEMBL29756362 0.65 KDM4E (0.51) ACHECYP1A2MAOAKDM4EALDH1A1
SCHEMBL29756454 0.63 DYRK1A (0.45) KDM4EALDH1A1HPGDGAA
SCHEMBL3461962 0.62 RXFP1 (0.41) HRH4KDM4EALDH1A1HPGDGAA
SCHEMBL29756406 0.61 PTPN5 (0.52) CYP1A2CYP2C19KDM4EALDH1A1HPGD
SCHEMBL20122732 0.61 PRKAB2 (0.48) ACHECYP1A2MAOAKDM4EALDH1A1
SCHEMBL29756387 0.61 CHEK2 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110382496-B Substituted pyrido [3,4-b ] indoles for the treatment of cartilage disorders 赛诺菲 2022-08-09 CN disclosed