SCHEMBL29759291

SCHEMBL29759291

CC(C)(C)OC(=O)N1CC(F)(F)CC1c1cc(F)cc(C(=O)O)c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 6/20 0.35
PDE5A O76074 3/20 0.34
P2RY14 Q15391 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
RIPK1 Q13546 2/20 0.33
JAK2 O60674 1/20 0.33
NTRK1 P04629 1/20 0.33
HCAR1 Q9BXC0 1/20 0.32
NR1H2 P55055 3/20 0.32
NR1H3 Q13133 3/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ROCK2 O75116 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24526756 1.00 TACR1 (0.35) TACR1PDE5AP2RY14HDAC1HDAC6
SCHEMBL24527025 0.89 UCHL1 (0.38) TACR1HDAC1HDAC6HDAC5RIPK1
SCHEMBL24527120 0.84 MMP9 (0.37) ROCK2
SCHEMBL12477897 0.83 AR (0.36) TACR1RIPK1NR1H2NR1H3
SCHEMBL456786 0.83 AR (0.36) TACR1RIPK1NR1H2NR1H3
SCHEMBL24526992 0.82 MMP9 (0.33) TACR1JAK2NTRK1ROCK2
SCHEMBL451781 0.82 RIPK1 (0.50) TACR1PDE5ARIPK1JAK2NTRK1
SCHEMBL21723215 0.82 RIPK1 (0.50) TACR1PDE5ARIPK1JAK2NTRK1
SCHEMBL29744544 0.82 RIPK1 (0.50) TACR1PDE5ARIPK1JAK2NTRK1
SCHEMBL430829 0.82 RIPK1 (0.50) TACR1PDE5ARIPK1JAK2NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129047-A2 NOVEL MODULATORS OF THE NMDA RECEPTOR H. LUNDBECK A/S (DK) 2022-06-23 WO disclosed