SCHEMBL29778034

SCHEMBL29778034

CC1(C)OB(c2ccc(C(F)(F)F)c3ncccc23)OC1(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
TNF P01375 1/20 0.38
CXCL8 P10145 1/20 0.38
KMT2A Q03164 1/20 0.38
PAX8 Q06710 1/20 0.38
KLF5 Q13887 1/20 0.38
NCF1 P14598 1/20 0.38
PARP1 P09874 1/20 0.38
SLC40A1 Q9NP59 3/20 0.36
KDM4E B2RXH2 2/20 0.35
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
NPC1 O15118 1/20 0.34
HSP90AA1 P07900 1/20 0.34
EPHX2 P34913 1/20 0.34
LIPE Q05469 3/20 0.34
GSK3A P49840 2/20 0.33
GSK3B P49841 2/20 0.33
DYRK3 O43781 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30018309 0.90 SLC40A1 (0.41) MEN1TNFCXCL8KMT2APAX8
SCHEMBL4013608 0.90 NCF1 (0.44) MEN1TNFCXCL8KMT2APAX8
SCHEMBL26922460 0.83 KDM4E (0.44) SLC40A1KDM4EL3MBTL1NPC1HSP90AA1
SCHEMBL29734917 0.83 KDM4E (0.44) SLC40A1KDM4EL3MBTL1NPC1HSP90AA1
SCHEMBL26921493 0.82 LIPE (0.38) SLC40A1KDM4EL3MBTL1NPC1HSP90AA1
SCHEMBL795284 0.81 MEN1 (0.43) MEN1KMT2ASLC40A1KDM4EL3MBTL1
SCHEMBL26920675 0.80 KDM4E (0.41) MEN1KMT2AKDM4EL3MBTL1NPC1
SCHEMBL26921299 0.80 L3MBTL1 (0.33) KDM4EL3MBTL1NPC1HSP90AA1MPI
SCHEMBL25216841 0.78 L3MBTL1 (0.49) MEN1KMT2ASLC40A1KDM4EL3MBTL1
SCHEMBL26920096 0.77 COMT (0.37) KMT2AKDM4EL3MBTL1NPC1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4039685-A1 AZABICYCLIC SHP2 INHIBITORS IRBM S.P.A. (IT) 2022-08-10 EP disclosed