SCHEMBL29787346

SCHEMBL29787346

CCCCn1cc2c(n1)c(Cl)nc1ccccc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.72
TLR7 Q9NYK1 1/20 0.72
SLC2A1 P11166 3/20 0.41
MPO P05164 3/20 0.41
MEN1 O00255 2/20 0.40
CYP1A2 P05177 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
KDM4E B2RXH2 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
ADORA3 P0DMS8 2/20 0.38
ADORA2A P29274 2/20 0.38
HTR4 Q13639 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
PDE4A P27815 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22806917 1.00 TLR8 (0.72) TLR8TLR7SLC2A1MPOMEN1
SCHEMBL5506468 0.92 TLR7 (0.60) TLR8TLR7SLC2A1MEN1KMT2A
SCHEMBL1233701 0.84 TLR8 (1.00) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL29720427 0.84 TLR8 (1.00) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL22445125 0.82 TLR8 (0.50) TLR8TLR7CYP1A2KDM4EALDH1A1
SCHEMBL17083434 0.78 MAOA (0.46) TLR8TLR7MEN1KMT2AKDM4E
SCHEMBL5507108 0.76 TLR7 (0.57) TLR8TLR7SLC2A1MEN1KMT2A
SCHEMBL1232530 0.75 TLR7 (0.85) TLR8TLR7ADORA3ADORA2AADORA1
SCHEMBL14323257 0.74 ADORA3 (0.48) TLR8TLR7CYP1A2KMT2AMAPT
SCHEMBL5507105 0.74 TLR8 (0.41) TLR8TLR7SLC2A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114746420-A 1- (4- (aminomethyl) benzyl) -2-butyl-2H-pyrazolo [3,4-c ] quinolin-4-amine derivatives as Toll-like receptor (TLR)7/8 agonists and related compounds and antibody drug conjugates thereof for cancer therapy and diagnosis 苏特罗生物制药公司 2022-07-12 CN disclosed