SCHEMBL2979402

SCHEMBL2979402

C=Cc1nccc(-c2cccnc2)c1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.45
GLA P06280 3/20 0.45
GAA P10253 3/20 0.45
CYP11B2 P19099 4/20 0.43
ADORA2A P29274 2/20 0.42
ADORA1 P30542 2/20 0.42
IKBKB O14920 1/20 0.41
NUDT1 P36639 1/20 0.41
ALDH1A1 P00352 4/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
RXFP1 Q9HBX9 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPK1 P28482 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
HPGD P15428 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2977681 0.85 ALDH1A1 (0.55) KDM4EGAAADORA2AADORA1ALDH1A1
SCHEMBL9697450 0.77 SMN1; SMN2 (0.47) KDM4EGLAGAACYP11B2ADORA2A
SCHEMBL30804680 0.75 ALDH1A1 (0.56) KDM4EGLAGAACYP11B2ADORA1
SCHEMBL2979399 0.74 ADORA2A (0.48) KDM4EGLAGAACYP11B2ADORA2A
SCHEMBL2974175 0.74 SQOR (0.41) KDM4EGLAGAAALDH1A1KMT2A
SCHEMBL30786742 0.73 ALDH1A1 (0.49) KDM4EGLAGAACYP11B2ADORA2A
SCHEMBL7100991 0.72 KDM4E (0.58) KDM4EGLAGAACYP11B2ADORA2A
SCHEMBL27756524 0.72 CYP2A6 (0.46) KDM4ECYP11B2NUDT1ALDH1A1CYP1A2
SCHEMBL16501607 0.71 NUDT1 (0.42) KDM4EGLAGAACYP11B2NUDT1
SCHEMBL28721464 0.71 KDM4E (0.50) KDM4EGLAGAACYP11B2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP disclosed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO disclosed