SCHEMBL297959

SCHEMBL297959

CCCCOC(=O)N1CCC(Oc2ncnc(N3CCc4cc(C(=O)O)ccc43)c2C)C(F)C1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 17/20 0.48
MAPT P10636 3/20 0.34
TP53 P04637 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298072 0.87 GPR119 (0.46) GPR119
SCHEMBL13034608 0.85 GPR119 (0.38) GPR119CYP2C9
SCHEMBL287664 0.82 GPR119 (0.37) GPR119CYP2C9
SCHEMBL298251 0.80 GPR119 (0.45) GPR119
SCHEMBL759241 0.79 GPR119 (0.36) GPR119CYP2C9
SCHEMBL3512362 0.71 GPR119 (0.36) GPR119CYP2C9
SCHEMBL757014 0.71 GPR119 (0.36) GPR119CYP2C9
SCHEMBL300080 0.71 GPR119 (0.36) GPR119CYP2C9
SCHEMBL290047 0.71 GPR119 (0.36) GPR119CYP2C9
SCHEMBL756660 0.70 GPR119 (0.35) GPR119CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427448-A1 Gpr 119 modulators Pfizer Inc. (US) 2012-03-14 EP disclosed
WO-2010128414-A1 GPR 119 MODULATORS PFIZER INC. (US) 2010-11-11 WO disclosed