SCHEMBL29796417

SCHEMBL29796417

c1cnc2ccc(-c3cnccn3)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 6/20 0.49
METAP2 P50579 1/20 0.45
CYP3A4 P08684 3/20 0.41
ALDH1A1 P00352 1/20 0.41
ADORA3 P0DMS8 1/20 0.39
DUSP4 Q13115 1/20 0.39
PTP4A1 Q93096 1/20 0.39
KCNH2 Q12809 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
CYP2A6 P11509 1/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PI4KA P42356 1/20 0.38
PIK3CG P48736 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29663058 0.84 ALDH1A1 (0.54) TGFBR1CYP3A4ALDH1A1KDM4EMAPT
Quinoline SCHEMBL9745228 0.81 ALDH1A1 (0.65) METAP2CYP3A4ALDH1A1DUSP4PTP4A1
SCHEMBL31418349 0.80 RAB9A (0.55) TGFBR1METAP2CYP3A4ALDH1A1DUSP4
SCHEMBL11992044 0.79 TGFBR1 (0.60) TGFBR1METAP2CYP3A4ALDH1A1KDM4E
SCHEMBL21352271 0.79 KDM4E (0.52) TGFBR1CYP3A4ALDH1A1KDM4EMAPT
Quinoline SCHEMBL29030603 0.76 ALDH1A1 (0.57) METAP2CYP3A4ALDH1A1DUSP4PTP4A1
SCHEMBL22824613 0.75 MIF (0.43) METAP2CYP3A4ALDH1A1DUSP4PTP4A1
SCHEMBL30433854 0.75 MIF (0.43) METAP2CYP3A4ALDH1A1DUSP4PTP4A1
SCHEMBL29661993 0.74 CCR1 (0.56) METAP2CYP3A4CYP2A6PIK3CDPIK3CA
SCHEMBL20169510 0.74 CCR1 (0.56) METAP2CYP3A4CYP2A6PIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728941-A Substituted 1, 5-naphthyridines or quinolines as ALK5 inhibitors 施万生物制药研发IP有限责任公司 2022-07-08 CN disclosed