SCHEMBL29802253

SCHEMBL29802253

CCOC(=O)c1cn(C2CC2)c2c(C)cc(F)cc2c1=O

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.57
KDM4E B2RXH2 3/20 0.44
KCNH2 Q12809 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP1A2 P05177 1/20 0.44
TOP2A P11388 5/20 0.44
TOP2B Q02880 5/20 0.44
STAT3 P40763 2/20 0.44
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10716822 0.89 ADRB2 (0.55) ADRB2KDM4EKCNH2SMN1; SMN2CYP1A2
SCHEMBL2844967 0.85 ADRB2 (0.68) ADRB2KDM4EKCNH2TOP2ATOP2B
SCHEMBL29492858 0.85 ADRB2 (0.68) ADRB2KDM4EKCNH2TOP2ATOP2B
SCHEMBL4713233 0.84 KDM4E (0.60) KDM4EKCNH2SMN1; SMN2CYP1A2TOP2A
SCHEMBL4564641 0.84 ADRB2 (0.57) ADRB2KDM4EKCNH2TOP2ATOP2B
SCHEMBL143605 0.83 ADRB2 (0.64) ADRB2KDM4EKCNH2TOP2ATOP2B
SCHEMBL3134035 0.83 ADRB2 (0.61) ADRB2KDM4EKCNH2TOP2ATOP2B
SCHEMBL10627001 0.83 ADRB2 (0.66) ADRB2KDM4EKCNH2TOP2ATOP2B
SCHEMBL8735574 0.83 ADRB2 (0.61) ADRB2KDM4EKCNH2TOP2ATOP2B
SCHEMBL7599453 0.82 ADRB2 (0.65) ADRB2KDM4EKCNH2TOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929224-A Novel medicine for treating hepatic encephalopathy 大塚制药株式会社 2022-08-19 CN disclosed