SCHEMBL29802408

SCHEMBL29802408

CSc1ccc(-c2cccc(Br)n2)cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.36
CYP2A6 P11509 1/20 0.36
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
SCN9A Q15858 1/20 0.34
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR7 P34969 1/20 0.33
NPC1 O15118 3/20 0.33
PKM P14618 3/20 0.33
RAB9A P51151 3/20 0.33
HSP90AA1 P07900 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA3 P34903 1/20 0.33
GRM5 P41594 2/20 0.32
TGFBR1 P36897 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23093432 1.00 HDAC1 (0.36) HDAC1CYP2A6PIK3CAMTORSCN9A
SCHEMBL31504097 0.81 CYP19A1 (0.45) CYP2A6NPC1RAB9AGABRA1GABRG2
SCHEMBL20390600 0.81 ASIC3 (0.49) HDAC1CYP2A6PIK3CAMTORSCN9A
SCHEMBL29802385 0.76 ALDH1A3 (0.42) NPC1RAB9AMAPK14MAPTALDH1A1
SCHEMBL23093241 0.76 ALDH1A3 (0.42) NPC1RAB9AMAPK14MAPTALDH1A1
SCHEMBL23093224 0.73 PIK3CD (0.43) CYP19A1
SCHEMBL29802465 0.73 PIK3CD (0.43) CYP19A1
SCHEMBL1334170 0.71 HSP90AA1 (0.53) HDAC1NPC1RAB9AHSP90AA1TGFBR1
SCHEMBL1404138 0.70
SCHEMBL28670824 0.67 RAB9A (0.62) NPC1PKMRAB9AHSP90AA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4027993-A1 CYCLOOXYGENASE-2 INHIBITORS AND USES THEREOF The Broad Institute Inc. (US) 2022-07-20 EP disclosed