SCHEMBL29802465

SCHEMBL29802465

CS(=O)(=O)c1ccc(-c2cccc(Br)n2)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.43
PIP5K1C O60331 1/20 0.43
PIK3CB P42338 1/20 0.43
PI4KA P42356 1/20 0.43
PIK3CG P48736 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
FAAH O00519 1/20 0.40
RORC P51449 1/20 0.37
ALOX5AP P20292 1/20 0.36
PLCG1 P19174 1/20 0.35
CYP19A1 P11511 2/20 0.34
LRRK2 Q5S007 1/20 0.34
ATR Q13535 3/20 0.33
GPR119 Q8TDV5 2/20 0.33
PDE10A Q9Y233 1/20 0.33
KCNH2 Q12809 1/20 0.33
PRKDC P78527 2/20 0.33
ATM Q13315 2/20 0.33
KCNJ1 P48048 1/20 0.32
TNF P01375 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23093224 1.00 PIK3CD (0.43) PIK3CDPIP5K1CPIK3CBPI4KAPIK3CG
SCHEMBL31504097 0.79 CYP19A1 (0.45) CYP19A1
SCHEMBL29802445 0.79 PTGS2 (0.48)
SCHEMBL23093438 0.79 PTGS2 (0.48)
SCHEMBL26107943 0.77 PI4KB (0.55) PIK3CDPIP5K1CPIK3CBPI4KAPIK3CG
SCHEMBL1404067 0.74 LOX (0.41) PLCG1
SCHEMBL30253017 0.74 LOX (0.41) PLCG1
SCHEMBL29802408 0.73 HDAC1 (0.36) CYP19A1
SCHEMBL23093432 0.73 HDAC1 (0.36) CYP19A1
SCHEMBL5700356 0.73 RORC (0.53) PIK3CDPIP5K1CPIK3CBPI4KAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4027993-A1 CYCLOOXYGENASE-2 INHIBITORS AND USES THEREOF The Broad Institute Inc. (US) 2022-07-20 EP disclosed