SCHEMBL29802440

SCHEMBL29802440

COCCOc1ncc(Br)nc1-c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.46
PTGS1 P23219 3/20 0.40
KCNH2 Q12809 2/20 0.39
LRRK2 Q5S007 1/20 0.39
CDK1 P06493 2/20 0.36
CDK2 P24941 2/20 0.36
KDR P35968 1/20 0.36
CCR4 P51679 1/20 0.36
ATR Q13535 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23093235 1.00 PTGS2 (0.46) PTGS2PTGS1KCNH2LRRK2CDK1
SCHEMBL29802518 0.86 PTGS2 (0.42) PTGS2PTGS1CDK1CDK2KDR
SCHEMBL23093191 0.86 PTGS2 (0.42) PTGS2PTGS1CDK1CDK2KDR
SCHEMBL23093139 0.85 LRRK2 (0.48) PTGS2PTGS1KCNH2LRRK2CCR4
SCHEMBL3816857 0.82 ALDH1A1 (0.40) CCR4
SCHEMBL23111085 0.80 EDNRB (0.36)
SCHEMBL29802439 0.80 PTGS2 (0.43) PTGS2PTGS1KCNH2LRRK2
SCHEMBL23093381 0.80 PTGS2 (0.43) PTGS2PTGS1KCNH2LRRK2
SCHEMBL23093419 0.76 KCNH2 (0.56) KCNH2ATR
SCHEMBL29802464 0.76 KCNH2 (0.56) KCNH2ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4027993-A1 CYCLOOXYGENASE-2 INHIBITORS AND USES THEREOF The Broad Institute Inc. (US) 2022-07-20 EP disclosed