SCHEMBL29802445

SCHEMBL29802445

CS(=O)(=O)c1ccc(-c2cccc(Br)n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.48
HDAC6 Q9UBN7 1/20 0.47
PTGS1 P23219 1/20 0.43
SCD O00767 1/20 0.42
GRM2 Q14416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23093438 1.00 PTGS2 (0.48) PTGS2HDAC6PTGS1SCDGRM2
SCHEMBL19243065 0.81 THRB (0.54) PTGS2HDAC6
SCHEMBL19237521 0.80 HDAC6 (0.44) PTGS2HDAC6PTGS1
SCHEMBL15730486 0.80 PTGS2 (0.48) PTGS2HDAC6PTGS1
SCHEMBL29802549 0.79 ASIC3 (0.56) PTGS2HDAC6
SCHEMBL23093295 0.79 PTGS2 (0.49) PTGS2HDAC6PTGS1
SCHEMBL29802375 0.79 PTGS2 (0.49) PTGS2HDAC6PTGS1
SCHEMBL23093471 0.79 ASIC3 (0.56) PTGS2HDAC6
SCHEMBL23093224 0.79 PIK3CD (0.43)
SCHEMBL29802465 0.79 PIK3CD (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4027993-A1 CYCLOOXYGENASE-2 INHIBITORS AND USES THEREOF The Broad Institute Inc. (US) 2022-07-20 EP disclosed