SCHEMBL29809376

SCHEMBL29809376

Nc1nc2ncccc2c2[nH]cnc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.42
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
PDPK1 O15530 1/20 0.39
GDA Q9Y2T3 1/20 0.39
PARP1 P09874 1/20 0.38
BRD4 O60885 1/20 0.38
ACHE P22303 2/20 0.38
NUDT1 P36639 1/20 0.38
PI4KA P42356 2/20 0.36
PI4K2B Q8TCG2 2/20 0.36
PI4K2A Q9BTU6 2/20 0.36
PI4KB Q9UBF8 2/20 0.36
LMNA P02545 1/20 0.36
DRD3 P35462 1/20 0.36
XDH P47989 1/20 0.36
LRRK2 Q5S007 1/20 0.36
HCAR2 Q8TDS4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1140927 1.00 DHFR (0.42) DHFRPDE4APDE4BPDE4CPDE4D
SCHEMBL212131 0.77 TLR7 (0.44) PDE4DPDPK1PARP1ACHENUDT1
SCHEMBL29694218 0.77 TLR7 (0.44) PDE4DPDPK1PARP1ACHENUDT1
SCHEMBL1007376 0.75 DHFR (0.53) DHFRPARP1ACHENUDT1LMNA
SCHEMBL30413516 0.75 PRMT5 (0.42) DHFRPDE4APDE4BPDE4CPDE4D
SCHEMBL311681 0.75 PRMT5 (0.42) DHFRPDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL5523405 0.75 RAB9A (0.44) PDE4DPDPK1PARP1ACHENUDT1
SCHEMBL4377817 0.75 DHFR (0.40) DHFRPARP1ACHENUDT1LMNA
Hydrochloric Acid SCHEMBL10587438 0.74 ALDH1A1 (0.46) PDE4DPDPK1PARP1ACHENUDT1
SCHEMBL28312743 0.73 TLR7 (0.44) PDE4DACHENUDT1LMNAADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805341-B Aromatic heterocyclic compound, and preparation method and application thereof 上海翊石医药科技有限公司 2023-12-08 CN disclosed
WO-2022161420-A1 CLASS OF HETEROAROMATIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海翊石医药科技有限公司 2022-08-04 WO disclosed
CN-114805341-A Aromatic heterocyclic compounds and preparation method and application thereof 上海翊石医药科技有限公司 2022-07-29 CN disclosed