SCHEMBL298304

SCHEMBL298304

O=C(O)c1cc2cccnc2n1-c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
TSHR P16473 1/20 0.45
PDE4B Q07343 9/20 0.42
ALKBH2 Q6NS38 1/20 0.41
EGLN1 Q9GZT9 1/20 0.41
DAO P14920 1/20 0.41
PDE4D Q08499 1/20 0.40
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MCL1 Q07820 1/20 0.40
NTRK1 P04629 1/20 0.39
NTRK3 Q16288 1/20 0.39
NAPRT Q6XQN6 1/20 0.39
P4HTM Q9NXG6 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9258763 0.84 ALDH1A1 (0.62) ALDH1A1TSHRALKBH2EGLN1DAO
SCHEMBL2539770 0.80 ALDH1A1 (0.54) ALDH1A1TSHRMEN1LMNAKMT2A
SCHEMBL297463 0.79 PDE4B (0.50) ALDH1A1TSHRPDE4BPDE4DMEN1
SCHEMBL296528 0.77 ALDH1A1 (0.47) ALDH1A1TSHRPDE4BPDE4DKDM4E
SCHEMBL28127748 0.75 KDM4E (0.44) ALDH1A1TSHRPDE4BDAOPDE4D
SCHEMBL3758947 0.75 MCL1 (0.56) ALDH1A1PDE4BDAOMEN1LMNA
SCHEMBL29904565 0.75 KDM4E (0.44) ALDH1A1TSHRPDE4BDAOPDE4D
SCHEMBL30226404 0.75 PARP1 (0.45) ALDH1A1TSHRPDE4BDAOPDE4D
SCHEMBL23672389 0.75 PDE4B (0.55) PDE4BPDE4D
SCHEMBL953080 0.75 KDM4E (0.43) ALDH1A1ALKBH2EGLN1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2106401-B1 DERIVATIVES OF PYRROLOPYRIDINE-2-CARBOXAMIDS, PREPARATION THEREOF AND THERAPEUTIC APPLICATION THEREOF SANOFI SA (FR) 2012-03-14 EP disclosed
EP-2106401-A2 DERIVATIVES OF PYRROLOPYRIDINE-2-CARBOXAMIDS, PREPARATION THEREOF AND THERAPEUTIC APPLICATION THEREOF Sanofi-Aventis (FR) 2009-10-07 EP disclosed
WO-2008107543-A2 DERIVATIVES OF PYRROLOPYRIDINE-2-CARBOXAMIDS, PREPARATION THEREOF AND THERAPEUTIC APPLICATION THEREOF SANOFI-AVENTIS (FR) 2008-09-12 WO disclosed