Myrophine

Myrophine

SCHEMBL29851007

CCCCCCCCCCCCCC(=O)O[C@H]1C=C[C@H]2[C@H]3Cc4ccc(OCc5ccccc5)c5c4[C@@]2(CCN3C)[C@H]1O5

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 10/20 0.56
OPRM1 P35372 12/20 0.56
OPRK1 P41145 10/20 0.56
MRGPRX2 Q96LB1 2/20 0.51
ADRB1 P08588 1/20 0.50
PDE4D Q08499 1/20 0.50
PDE3A Q14432 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Myrophine SCHEMBL26043 1.00 OPRD1 (0.56) OPRD1OPRM1OPRK1MRGPRX2ADRB1
SCHEMBL3477477 0.89 OPRM1 (0.71) OPRD1OPRM1OPRK1MRGPRX2ADRB1
SCHEMBL7775794 0.89 OPRM1 (0.71) OPRD1OPRM1OPRK1MRGPRX2ADRB1
SCHEMBL7770909 0.89 OPRM1 (0.71) OPRD1OPRM1OPRK1MRGPRX2ADRB1
SCHEMBL3477727 0.86 OPRM1 (0.73) OPRD1OPRM1OPRK1MRGPRX2ADRB1
SCHEMBL29610430 0.85 OPRM1 (0.77) OPRD1OPRM1OPRK1MRGPRX2ADRB1
SCHEMBL22959877 0.85 OPRM1 (0.77) OPRD1OPRM1OPRK1MRGPRX2ADRB1
SCHEMBL3477203 0.84 OPRM1 (0.70) OPRD1OPRM1OPRK1MRGPRX2ADRB1
SCHEMBL8208039 0.83 OPRM1 (0.62) OPRD1OPRM1OPRK1
SCHEMBL19463540 0.83 OPRD1 (0.72) OPRD1OPRM1OPRK1MRGPRX2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3064199-B1 ABUSE-DETERRENT TRANSDERMAL FORMULATIONS OF OPIATE AGONISTS AND AGONIST-ANTAGONISTS BUZZZ PHARMACEUTICALS LTD (IE) 2023-12-20 EP claimed
EP-3313407-B1 TREATMENT AND MANAGEMENT OF AUGMENTATION IN RESTLESS LEGS SYNDROME UNIV EAST CAROLINA (US) 2023-07-19 EP claimed
EP-3385252-B1 CANNABINOID RECEPTOR MODULATORS ARENA PHARM INC (US) 2022-09-21 EP claimed
EP-3291676-B1 MITRAGYNINE ANALOGS AND USES THEREOF MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-08-17 EP claimed
CN-113939277-B Formulations and methods for drug infusion into the bladder and treatment of bladder diseases 特瑞纲制药有限公司 2024-04-09 CN disclosed
CN-117295508-A Opioid dosage reduction compositions and methods of use thereof 迈索布拉斯特国际有限公司 2023-12-26 CN disclosed
EP-1765303-B2 ORAL TABLET SAFEGUARDED AGAINST ABUSE GRUENENTHAL GMBH (DE) 2022-11-23 EP disclosed