SCHEMBL29867907

SCHEMBL29867907

NC(=O)c1c2n(ccc1=O)CCOC2

nearest known ligand 0.30

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.30
HTT P42858 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30791523 0.80 KDM4E (0.38) KDM4EHTTALDH1A1
SCHEMBL15157482 0.71 HTT (0.37) HTT
SCHEMBL29867991 0.71 ALDH1A1 (0.34) KDM4EHTTALDH1A1
SCHEMBL30174263 0.69 ALOX5 (0.39) KDM4EHTTALDH1A1
SCHEMBL30174183 0.69 RIPK1 (0.35)
SCHEMBL30174188 0.68 TSHR (0.45) KDM4EALDH1A1
SCHEMBL30174220 0.68 CSNK1E (0.38) ALDH1A1
SCHEMBL17574521 0.67 KCNK3 (0.43) KDM4EALDH1A1
SCHEMBL15166031 0.67 ABCB1 (0.38) KDM4EALDH1A1
SCHEMBL30293754 0.66 AKR1C3 (0.38) KDM4EHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4294804-B1 PYRIDONE COMPOUNDS AND METHODS OF USE EXELIXIS INC (US) 2026-04-08 EP claimed
EP-4294804-A1 PYRIDONE COMPOUNDS AND METHODS OF USE Exelixis, Inc. (US) 2023-12-27 EP claimed
WO-2022178205-A1 PYRIDONE COMPOUNDS AND METHODS OF USE EXELIXIS, INC. (US) 2022-08-25 WO claimed
CN-117440951-A Pyridone compounds and methods of use 埃克塞里艾克西斯公司 2024-01-23 CN disclosed
EP-4294804-A1 PYRIDONE COMPOUNDS AND METHODS OF USE Exelixis, Inc. (US) 2023-12-27 EP disclosed
WO-2022178205-A1 PYRIDONE COMPOUNDS AND METHODS OF USE EXELIXIS, INC. (US) 2022-08-25 WO disclosed