SCHEMBL29888798

SCHEMBL29888798

COCCOc1ccc(Br)cc1CN(C)C

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.57
SLC6A4 P31645 7/20 0.50
SLC6A2 P23975 5/20 0.50
SLC6A3 Q01959 2/20 0.50
KMT2A Q03164 3/20 0.41
LMNA P02545 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
KDM4E B2RXH2 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
HPGD P15428 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 2/20 0.40
POLB P06746 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29888844 0.81 SLC6A4 (0.56) CCR5SLC6A4SLC6A2SLC6A3KMT2A
SCHEMBL3696560 0.81 SLC6A4 (0.56) CCR5SLC6A4SLC6A2SLC6A3KMT2A
SCHEMBL1516692 0.79 FBP1 (0.44) SLC6A4KMT2ALMNASMN1; SMN2KDM4E
SCHEMBL31053304 0.79 FBP1 (0.44) SLC6A4KMT2ALMNASMN1; SMN2KDM4E
SCHEMBL29964333 0.79 CCR5 (0.52) CCR5SLC6A4SLC6A2SLC6A3KMT2A
SCHEMBL29965019 0.76 CCR5 (0.56) CCR5SLC6A4SLC6A2SLC6A3KMT2A
SCHEMBL425797 0.76 FBP1 (0.48) KMT2ASMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL858361 0.76 FDPS (0.50) KMT2ASMN1; SMN2KDM4ENPC1RAB9A
SCHEMBL4573266 0.76 KDM4E (0.58) KMT2ALMNASMN1; SMN2KDM4ERAB9A
SCHEMBL4641066 0.75 KDM4E (0.48) KMT2ALMNASMN1; SMN2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022171034-A1 BICYCLIC COMPOUND AS HPK1 INHIBITOR AND APPLICATION THEREOF 江苏先声药业有限公司 2022-08-18 WO disclosed