SCHEMBL298910

SCHEMBL298910

CCC(c1ccc(C(N)=O)cc1C(=O)c1c[nH]c2ncccc12)S(=O)(=O)O

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 3/20 0.44
MAP2K1 Q02750 1/20 0.42
NEK2 P51955 2/20 0.42
KDR P35968 1/20 0.39
GRM8 O00222 1/20 0.38
GRM4 Q14833 1/20 0.38
HAT1 O14929 1/20 0.37
EP300 Q09472 1/20 0.37
ADORA2A P29274 1/20 0.35
MTNR1A P48039 1/20 0.35
CNR2 P34972 1/20 0.35
BRAF P15056 1/20 0.35
PRKCI P41743 1/20 0.34
CCNE1 P24864 3/20 0.34
CDK2 P24941 3/20 0.34
PKM P14618 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL297658 0.87 DYRK1A (0.43) CAMKK2NEK2KDRCDK2MKNK1
SCHEMBL299284 0.85 BRAF (0.45) CAMKK2MAP2K1NEK2KDRBRAF
SCHEMBL298640 0.85 BRAF (0.37) CAMKK2MAP2K1NEK2KDRBRAF
SCHEMBL297931 0.81 BRAF (0.43) CAMKK2MAP2K1NEK2KDRHAT1
SCHEMBL298168 0.80 PAK1 (0.49) MKNK1MKNK2
SCHEMBL299033 0.78 BRAF (0.46) MAP2K1NEK2KDRBRAFPKM
SCHEMBL3711232 0.76 CAMKK2 (0.54) CAMKK2MAP2K1NEK2KDRADORA2A
SCHEMBL3709076 0.73 NEK2 (0.63) CAMKK2MAP2K1NEK2KDRADORA2A
SCHEMBL298411 0.73 PAK1 (0.48) MKNK1MKNK2
SCHEMBL297872 0.72 CYP2C9 (0.48) MAP2K1NEK2KDRBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed