SCHEMBL29891817

SCHEMBL29891817

Cc1ccccc1-n1cc(C2CCN(C(=O)OC(C)(C)C)CC2)cn1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
TP53 P04637 6/20 0.51
MAPT P10636 4/20 0.51
LMNA P02545 4/20 0.51
GRM5 P41594 1/20 0.49
GRM1 Q13255 1/20 0.49
NAMPT P43490 1/20 0.48
THRB P10828 2/20 0.47
POLB P06746 1/20 0.46
GPR119 Q8TDV5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23410880 1.00 MEN1 (0.51) MEN1KMT2ATP53MAPTLMNA
SCHEMBL25168756 0.84 HSD11B1 (0.47) KMT2ATP53MAPTLMNA
SCHEMBL20135488 0.83 GPR119 (0.58) MEN1KMT2ATP53MAPTLMNA
SCHEMBL23411297 0.81 GRM5 (0.62) MEN1KMT2ATP53MAPTLMNA
SCHEMBL23411546 0.80 MGLL (0.51) MEN1KMT2ATP53MAPTLMNA
SCHEMBL32661690 0.79 GPR119 (0.56) MEN1KMT2ATP53MAPTNAMPT
SCHEMBL4473713 0.78 THRB (0.50) MEN1KMT2ATP53MAPTNAMPT
SCHEMBL30795957 0.78 PBRM1 (0.67) MEN1KMT2A
SCHEMBL25794242 0.77 MEN1 (0.52) MEN1KMT2ATP53MAPTLMNA
SCHEMBL18866042 0.77 GPR119 (0.48) MEN1KMT2ATP53LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119564686-A DGK alpha inhibitors as immune activation substituted aminoquinolones of (2) 拜耳公司 2025-03-07 CN disclosed
CN-119523983-A DGK alpha inhibitors as immune activation substituted aminoquinolones of (2) 拜耳公司 2025-02-28 CN disclosed
CN-119424429-A DGK alpha inhibitors as immune activation substituted aminoquinolones of (2) 拜耳公司 2025-02-14 CN disclosed
CN-115003665-B DGK alpha inhibitors as immune activation substituted aminoquinolones of (2) 拜耳公司 2024-11-08 CN disclosed
EP-4065574-A1 SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION Bayer Aktiengesellschaft (DE) 2022-10-05 EP disclosed
CN-115003665-A Substituted aminoquinolones as immunoactive DGK alpha inhibitors 拜耳公司 2022-09-02 CN disclosed