SCHEMBL29893282

SCHEMBL29893282

N=CC1c2ccccc2-c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 2/20 0.41
HTR2A P28223 2/20 0.41
POLB P06746 2/20 0.39
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
ACHE P22303 3/20 0.33
BCHE P06276 2/20 0.33
S100A4 P26447 1/20 0.33
CHRM2 P08172 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19973035 1.00 GPR3 (0.41) GPR3HTR2APOLBHDAC3HDAC4
Toluene SCHEMBL28351667 0.87 LMNA (0.44) GPR3HTR2APOLBKMT2AACHE
SCHEMBL6421466 0.78 GPR3 (0.44) GPR3HTR2APOLBHDAC3HDAC4
SCHEMBL29711937 0.74 GPR3 (0.41) GPR3HTR2APOLBHDAC3HDAC4
SCHEMBL1766205 0.74 GPR3 (0.46) GPR3HTR2APOLBHDAC3HDAC4
SCHEMBL1568290 0.74 GPR3 (0.46) GPR3HTR2APOLBHDAC3HDAC4
SCHEMBL224931 0.74 GPR3 (0.41) GPR3HTR2APOLBHDAC3HDAC4
SCHEMBL1766128 0.74 GPR3 (0.41) GPR3HTR2APOLBHDAC3HDAC4
SCHEMBL7421342 0.74 GPR3 (0.41) GPR3HTR2APOLBHDAC3HDAC4
SCHEMBL29196425 0.74 GPR3 (0.41) GPR3HTR2APOLBHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4294392-A1 TARGETED BIFUNCTIONAL DEGRADERS AND METHODS USING SAME Yale University, Inc. (US) 2023-12-27 EP disclosed
WO-2022178428-A1 TARGETED BIFUNCTIONAL DEGRADERS AND METHODS USING SAME YALE UNIVERSITY (US) 2022-08-25 WO disclosed