SCHEMBL29907301

SCHEMBL29907301

COC(=O)Cc1cccc2c1ncn2COCC[Si](C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.38
DGAT1 O75907 3/20 0.36
NPC1 O15118 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
KDM4E B2RXH2 1/20 0.34
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
EPHB4 P54760 1/20 0.32
TEK Q02763 1/20 0.32
ICMT O60725 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27139837 1.00 KMT2A (0.38) KMT2ADGAT1NPC1ADORA2AADORA1
SCHEMBL22717563 0.83 NPC1 (0.37) KMT2ADGAT1NPC1ADORA2AADORA1
SCHEMBL29117045 0.82 EGLN3 (0.36) DGAT1NPC1ADORA2AADORA1MAPT
SCHEMBL27142590 0.82 DGAT1 (0.36) KMT2ADGAT1NPC1KDM4EMTNR1A
SCHEMBL30897282 0.82 DGAT1 (0.36) KMT2ADGAT1NPC1KDM4EMTNR1A
SCHEMBL22717628 0.82 ALDH1A1 (0.38) KMT2ADGAT1NPC1KDM4EMAPT
SCHEMBL27251064 0.78 CYP17A1 (0.38) DGAT1NPC1KDM4EBRD4CREBBP
SCHEMBL4006680 0.77 EGFR (0.44) KMT2ADGAT1NPC1KDM4EEGFR
SCHEMBL5951884 0.77 DGAT1 (0.38) DGAT1NPC1BRD4CREBBPEGFR
SCHEMBL29907237 0.77 NPC1 (0.34) KMT2ADGAT1NPC1BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4602047-A1 THIAZOLO[5,4-D]PYRIMIDINE COMPOUNDS, COMPOSITIONS COMPRISING THEM AND USES THEREOF The Universite de Montreal (CA) 2025-08-20 EP disclosed
WO-2024077391-A1 THIAZOLO[5,4-D]PYRIMIDINE COMPOUNDS, COMPOSITIONS COMPRISING THEM AND USES THEREOF UNIVERSITE DE MONTREAL (CA) 2024-04-18 WO disclosed
EP-4326719-A1 PYRIDO[3,2-D]PYRIMIDINE COMPOUNDS USES THEREOF FOR TREATING A PROLIFERATIVE DISEASE Université de Montréal (CA) 2024-02-28 EP disclosed
WO-2022221939-A1 PYRIDO[3,2-D]PYRIMIDINE COMPOUNDS USES THEREOF FOR TREATING A PROLIFERATIVE DISEASE UNIVERSITE DE MONTREAL (CA) 2022-10-27 WO disclosed