SCHEMBL29907659

SCHEMBL29907659

Cn1cc(-c2nc(C(N)=O)cnc2-c2ccc(F)cc2)ccc1=O

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.56
ADORA1 P30542 8/20 0.56
BRD4 O60885 1/20 0.50
CREBBP Q92793 1/20 0.43
ADORA2B P29275 7/20 0.41
MAPK1 P28482 1/20 0.41
CNR1 P21554 2/20 0.40
ADORA3 P0DMS8 1/20 0.39
TGFBR1 P36897 3/20 0.39
TGFBR2 P37173 2/20 0.39
NPY5R Q15761 1/20 0.38
TNIK Q9UKE5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585799 0.83 ADORA2A (0.75) ADORA2AADORA1BRD4CREBBPADORA2B
SCHEMBL29907731 0.80 ADORA2A (0.52) ADORA2AADORA1ADORA2BCNR1ADORA3
SCHEMBL29907757 0.80 ADORA2A (0.48) ADORA2AADORA1BRD4ADORA2BCNR1
SCHEMBL29907672 0.80 ADORA2A (0.51) ADORA2AADORA1BRD4ADORA2B
SCHEMBL4585557 0.80 ADORA2A (0.65) ADORA2AADORA1BRD4CREBBPADORA2B
SCHEMBL29907681 0.79 ADORA2A (0.48) ADORA2AADORA1BRD4CREBBPADORA2B
SCHEMBL29907708 0.78 TGFBR1 (0.51) ADORA2AADORA1TGFBR1TGFBR2
SCHEMBL29906682 0.77 ADORA2A (0.47) ADORA2AADORA1ADORA2BTGFBR1TGFBR2
SCHEMBL29907763 0.77 ADORA2A (0.47) ADORA2AADORA1ADORA2BTGFBR1TGFBR2
SCHEMBL29987316 0.75 ADORA2A (0.65) ADORA2AADORA1BRD4CREBBPADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed