SCHEMBL29907760

SCHEMBL29907760

Cc1cc(-c2nc(C(N)=O)cnc2-c2ncco2)cc(C)n1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 4/20 0.36
ADORA2A P29274 7/20 0.35
ADORA2B P29275 3/20 0.35
ADORA1 P30542 5/20 0.35
PIK3CB P42338 1/20 0.34
TGFBR1 P36897 2/20 0.34
DGAT1 O75907 2/20 0.34
SOAT1 P35610 1/20 0.34
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
CNR1 P21554 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
GLRA3 O75311 1/20 0.32
GLRB P48167 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29907672 0.79 ADORA2A (0.51) ADORA2AADORA2BADORA1
SCHEMBL29907604 0.77 ADORA2A (0.61) ADORA2AADORA2BADORA1TGFBR1
SCHEMBL29907731 0.74 ADORA2A (0.52) ADORA2AADORA2BADORA1DGAT1SOAT1
SCHEMBL29907725 0.74 ADORA2A (0.54) ADORA2AADORA2BADORA1
SCHEMBL29907696 0.73 ADORA2A (0.46) IRAK4ADORA2AADORA2BADORA1
SCHEMBL29907536 0.72 ADORA2A (0.49) ADORA2AADORA2BADORA1TGFBR1
SCHEMBL29907714 0.68 ADORA2A (0.51) ADORA2AADORA2BADORA1
SCHEMBL29906724 0.66 SIRT6 (0.44) GLRA3GLRB
SCHEMBL3347772 0.65 GLRA3 (0.44) PIK3CBTLR8CCNCCDK8GLRA3
SCHEMBL5554203 0.65 IL2 (0.46) TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed