SCHEMBL29908423

SCHEMBL29908423

O=C1NCC2COc3cccnc3N12

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.39
RIPK1 Q13546 11/20 0.36
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
MAPK1 P28482 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
PDE3A Q14432 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
LTA4H P09960 5/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29908470 0.82 NOTUM (0.42) NR3C2RIPK1LTA4H
SCHEMBL29908458 0.78 PARP1 (0.39) NR3C2RIPK1ALDH1A1LMNAPOLB
SCHEMBL7471047 0.77 NOTUM (0.43) ALDH1A1LMNALTA4H
SCHEMBL29908490 0.76 RIPK1 (0.38) NR3C2RIPK1LTA4H
SCHEMBL26914996 0.71 HTR2A (0.58)
SCHEMBL31022150 0.71 HTR2A (0.58)
SCHEMBL31022237 0.70 HTR2A (0.42) NR3C2
SCHEMBL4716719 0.70 CD74 (0.40) NR3C2ALDH1A1LMNAPOLBADORA3
SCHEMBL21807029 0.69 MEN1 (0.48) LTA4H
SCHEMBL21807075 0.69 MEN1 (0.48) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115028649-A Tricyclic compound, pharmaceutical composition containing same and use thereof 四川科伦博泰生物医药股份有限公司 2022-09-09 CN disclosed