SCHEMBL29912895

SCHEMBL29912895

FC(F)(F)c1cccc(-c2nc3ncc(Br)nc3[nH]2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.41
GABRG2 P18507 2/20 0.41
GABRB3 P28472 2/20 0.41
GABRA3 P34903 2/20 0.41
DGAT2 Q96PD7 3/20 0.41
IDH1 O75874 7/20 0.38
IDH2 P48735 2/20 0.38
METAP2 P50579 1/20 0.38
METAP1 P53582 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HTT P42858 2/20 0.37
KMT2A Q03164 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
HSP90AA1 P07900 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NOTUM Q6P988 1/20 0.36
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27158228 1.00 GABRA1 (0.41) GABRA1GABRG2GABRB3GABRA3DGAT2
SCHEMBL15922752 0.72 METAP2 (0.60) GABRA1GABRG2GABRB3GABRA3DGAT2
SCHEMBL29912896 0.71 PI4KA (0.46) ALDH1A1KMT2AMEN1HPGDSMN1; SMN2
SCHEMBL29202322 0.71 PI4KA (0.46) ALDH1A1KMT2AMEN1HPGDSMN1; SMN2
SCHEMBL29912851 0.69 GABRA1 (0.40) GABRA1GABRG2GABRB3GABRA3IDH1
SCHEMBL27157974 0.69 GABRA1 (0.40) GABRA1GABRG2GABRB3GABRA3IDH1
SCHEMBL29418961 0.69 NOTUM (0.41) GABRA1GABRG2GABRB3GABRA3DGAT2
SCHEMBL15094600 0.69 NOTUM (0.41) GABRA1GABRG2GABRB3GABRA3DGAT2
SCHEMBL15624402 0.67 NOTUM (0.58) GABRA1GABRG2GABRB3GABRA3IDH1
SCHEMBL30395354 0.67 NOTUM (0.58) GABRA1GABRG2GABRB3GABRA3IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4329881-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF Vanqua Bio, Inc. (US) 2024-03-06 EP disclosed
CN-117642404-A Small molecule modulators of glucocerebrosidase activity and uses thereof 凡况生化公司 2024-03-01 CN disclosed
WO-2022232383-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2022-11-03 WO disclosed