SCHEMBL29912896

SCHEMBL29912896

Brc1cnc2nc(-c3ccccc3)[nH]c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.46
PI4K2B Q8TCG2 1/20 0.46
PI4K2A Q9BTU6 1/20 0.46
PI4KB Q9UBF8 1/20 0.46
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GSK3B P49841 2/20 0.42
FGFR1 P11362 1/20 0.42
FGFR2 P21802 1/20 0.42
IKBKE Q14164 1/20 0.41
TBK1 Q9UHD2 1/20 0.41
NPY5R Q15761 1/20 0.41
SCN2A Q99250 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29202322 1.00 PI4KA (0.46) PI4KAPI4K2BPI4K2API4KBMEN1
SCHEMBL11829946 0.78 GAA (0.50) PI4KAPI4K2BPI4K2API4KBMEN1
SCHEMBL4046146 0.75 METAP2 (0.64) PI4KAPI4K2BPI4K2API4KBGSK3B
SCHEMBL11839052 0.74 ADORA3 (0.47) PI4KAPI4K2BPI4K2API4KBMEN1
SCHEMBL1667430 0.72 AURKA (0.68) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL5249728 0.72 GAA (0.53) PI4KAPI4K2BPI4K2API4KBMEN1
SCHEMBL29912895 0.71 GABRA1 (0.41) MEN1KMT2AALDH1A1HPGDSMN1; SMN2
SCHEMBL27158496 0.71 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2GSK3BIKBKETBK1
SCHEMBL22516593 0.69 SMN1; SMN2 (0.50) SMN1; SMN2
SCHEMBL23001457 0.69 NUDT1 (0.44) KMT2AALDH1A1MAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4329881-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF Vanqua Bio, Inc. (US) 2024-03-06 EP disclosed
CN-117642404-A Small molecule modulators of glucocerebrosidase activity and uses thereof 凡况生化公司 2024-03-01 CN disclosed
WO-2022232383-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2022-11-03 WO disclosed