SCHEMBL29923737

SCHEMBL29923737

COc1ccc(I)c2cc(C)cnc12

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.40
CCR5 P51681 1/20 0.40
CCR8 P51685 1/20 0.40
HPGDS O60760 1/20 0.38
ACHE P22303 1/20 0.37
MAPT P10636 1/20 0.37
POLB P06746 1/20 0.36
KAT2B Q92831 1/20 0.35
ATP4A P20648 2/20 0.35
ATP4B P51164 2/20 0.35
KIT P10721 1/20 0.35
NQO2 P16083 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP19A1 P11511 1/20 0.34
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24916302 1.00 CCR1 (0.40) CCR1CCR5CCR8HPGDSACHE
SCHEMBL24916307 0.83 CCR1 (0.42) CCR1CCR5CCR8HPGDSACHE
SCHEMBL24715886 0.80 NQO2 (0.47) CCR1CCR5CCR8HPGDSACHE
SCHEMBL24715871 0.80 CCR1 (0.40) CCR1CCR5CCR8HPGDSACHE
SCHEMBL24715864 0.80 MAPT (0.44) CCR1CCR5CCR8HPGDSACHE
SCHEMBL24916213 0.78 ATP4A (0.43) CCR1CCR5CCR8HPGDSACHE
SCHEMBL4414248 0.72 PDK2 (0.40) MAPTPOLBKITNQO2CYP19A1
SCHEMBL434888 0.69 HPGDS (0.62) CCR1CCR5CCR8HPGDSMAPT
SCHEMBL10112981 0.69 ACHE (0.43) CCR1CCR5CCR8ACHEMAPT
SCHEMBL16431498 0.67 MAPT (0.41) ACHEMAPTPOLBKAT2BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed