SCHEMBL29924550

SCHEMBL29924550

CC1(c2ccc(Cl)cc2F)C=CC=CC1

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.31
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29947353 1.00 KMT2A (0.31) KMT2ABACE1
SCHEMBL30404309 1.00 KMT2A (0.31) KMT2ABACE1
SCHEMBL31009242 0.79 PDE2A (0.36) BACE1
SCHEMBL31009251 0.79 TRPV4 (0.36) KMT2A
SCHEMBL30938761 0.78 CYP11B2 (0.38)
SCHEMBL29993382 0.75 PDK2 (0.31)
SCHEMBL30680744 0.74 SLC6A4 (0.33) BACE1
SCHEMBL30217567 0.73 MAPK1 (0.34) KMT2A
SCHEMBL29800290 0.72 CXCR3 (0.37) KMT2A
SCHEMBL14625577 0.71 PTGDR (0.37) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118344349-A 4-Alkoxybenzimidazole-6-carboxylic acid derivatives as GLP-1 receptor agonists 中国科学院上海药物研究所 2024-07-16 CN disclosed
CN-113853371-B GLP-1R agonists and uses thereof 上海齐鲁锐格医药研发有限公司 2024-05-03 CN disclosed
EP-4334304-A1 BENZIMIDAZOYL GLP-1 RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME, AND METHODS FOR THEIR USE Carmot Therapeutics, Inc. (US) 2024-03-13 EP disclosed
CN-117279904-A GLP-1 receptor agonists, pharmaceutical compositions comprising same and methods of making same 株式会社LG化学 2023-12-22 CN disclosed
CN-117222644-A 2- ((4- ((S) -2- (4-chloro-2-fluorophenyl) -2-methylbenzo [ d ] [1,3] dioxol-4-yl) piperidin-1-yl) methyl) -1- (((S) -oxetan-2-yl) methyl) -1H-imidazole derivatives as GLP1 receptor activators for the treatment of obesity 诺华股份有限公司 2023-12-12 CN disclosed
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
CN-116547278-A Heterocyclic GLP-1 agonists 加舒布鲁姆生物公司 2023-08-04 CN disclosed
CN-116323599-A Heterocyclic GLP-1 agonists 加舒布鲁姆生物公司 2023-06-23 CN disclosed
CN-116217558-A GLP-1 receptor agonist, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2023-06-06 CN disclosed
CN-115667250-A Heterocyclic GLP-1 agonists 加舒布鲁姆生物公司 2023-01-31 CN disclosed
CN-115521297-A 5,6-dihydro-1,2,4-triazines and their pharmaceutical use as GLP-1 receptor agonists 中国科学院上海药物研究所 2022-12-27 CN disclosed
CN-115335374-A GLP-1R modulating compounds 吉利德科学公司 2022-11-11 CN disclosed
WO-2022235717-A1 BENZIMIDAZOYL GLP-1 RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME, AND METHODS FOR THEIR USE CARMOT THERAPEUTICS, INC. (US) 2022-11-10 WO disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed