SCHEMBL29924912

SCHEMBL29924912

CCOC(=O)c1cc2c(nc(C)n2CCOC)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.44
TSHR P16473 3/20 0.44
GAA P10253 3/20 0.44
PTGER4 P35408 3/20 0.42
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 4/20 0.39
CASP7 P55210 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
HPGD P15428 2/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
RECQL P46063 1/20 0.39
RAB9A P51151 1/20 0.39
ESR2 Q92731 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
USP2 O75604 1/20 0.39
GLA P06280 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29924614 0.90 CSNK2A2 (0.42) HSD17B10TSHRGAAPTGER4KDM4E
SCHEMBL29924734 0.86 HSD17B10 (0.41) HSD17B10TSHRGAAPTGER4KDM4E
SCHEMBL29149723 0.86 DAPK3 (0.41) PTGER4KDM4EALDH1A1L3MBTL1HPGD
SCHEMBL6306238 0.79 MAPT (0.38) HSD17B10TSHRGAAKDM4EALDH1A1
SCHEMBL6774504 0.77 HSD17B10 (0.42) HSD17B10TSHRGAAKDM4EALDH1A1
SCHEMBL6300563 0.74 LMNA (0.52) GAAKDM4EALDH1A1L3MBTL1HPGD
SCHEMBL22677882 0.73 CYP3A4 (0.36) TSHRGAAKDM4EALDH1A1NPSR1
SCHEMBL27286488 0.72 HSD17B10 (0.43) HSD17B10TSHRGAAKDM4EALDH1A1
SCHEMBL24434035 0.71 PIK3CA (0.42) HSD17B10TSHRGAAKDM4EALDH1A1
SCHEMBL29149855 0.71 DAPK3 (0.36) PTGER4KDM4EALDH1A1L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed