SCHEMBL29926543

SCHEMBL29926543

Cc1c[nH]c2cccc(C(N)=O)c12

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
ATM Q13315 2/20 0.50
PARP1 P09874 6/20 0.47
GAA P10253 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
GPR84 Q9NQS5 1/20 0.42
NR4A2 P43354 1/20 0.42
BTK Q06187 4/20 0.41
PDPK1 O15530 1/20 0.41
CTNNB1 P35222 1/20 0.41
WNT3A P56704 1/20 0.41
PARP2 Q9UGN5 2/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2588267 1.00 ALDH1A1 (0.50) ALDH1A1ATMPARP1GAANPSR1
SCHEMBL2592748 0.84 HSD17B10 (0.47) ALDH1A1ATMPARP1GAAGPR84
SCHEMBL1223596 0.80 NR4A2 (0.61) ALDH1A1ATMNR4A2NPC1
SCHEMBL29886596 0.80 NR4A2 (0.61) ALDH1A1ATMNR4A2NPC1
SCHEMBL3721316 0.78 GPR84 (0.49) ALDH1A1ATMGAANPSR1GPR84
SCHEMBL15836985 0.78 TSHR (0.54) ALDH1A1GAANR4A2
SCHEMBL3960635 0.75 GPR84 (0.49) ALDH1A1ATMGAANPSR1GPR84
SCHEMBL3995494 0.74 GPR84 (0.51) ALDH1A1GAAGPR84NR4A2CTNNB1
SCHEMBL15356576 0.74 PBRM1 (0.56) ALDH1A1ATMGAAGPR84NR4A2
SCHEMBL16339986 0.74 ALDH1A1 (0.56) ALDH1A1ATMPARP1GAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117813095-A VCP inhibitors for the treatment of amyotrophic lateral sclerosis 弗朗西斯克里克研究所有限公司 2024-04-02 CN claimed
CN-117813095-A VCP inhibitors for the treatment of amyotrophic lateral sclerosis 弗朗西斯克里克研究所有限公司 2024-04-02 CN disclosed
CN-116947856-A EZH2 inhibitor and preparation method and application thereof 星希尔生物科技(上海)有限公司 2023-10-27 CN disclosed
CN-116768857-A EZH2/HDAC double-target inhibitor and preparation method and medical application thereof 中国药科大学 2023-09-19 CN disclosed
CN-112920176-B Bifunctional compound capable of inducing PRC2 protein complex core subunit degradation, pharmaceutical composition and application 四川大学华西医院 2022-11-04 CN disclosed