SCHEMBL29927588

SCHEMBL29927588

Nc1nc(N)n(-c2nccc3ccccc23)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AXL P30530 2/20 0.51
PLAU P00749 2/20 0.49
F12 P00748 2/20 0.49
NCF1 P14598 1/20 0.49
NOS3 P29474 1/20 0.49
NOS1 P29475 1/20 0.49
NOS2 P35228 1/20 0.49
BACE1 P56817 1/20 0.49
HRH4 Q9H3N8 1/20 0.45
HTR2C P28335 1/20 0.45
CYP2A6 P11509 1/20 0.41
COMT P21964 1/20 0.40
PLG P00747 1/20 0.38
SORD Q00796 2/20 0.38
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
F2 P00734 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12779077 0.79 AXL (0.71) AXLPLAUF12NCF1NOS3
SCHEMBL29928526 0.75 HTR2C (0.46) AXLHTR2CALDH1A1
SCHEMBL29928245 0.74 ATM (0.49) ALDH1A1MAPTRAB9ASMN1; SMN2ATM
SCHEMBL6086513 0.73 PLAU (0.47) AXLPLAUF12NCF1NOS3
SCHEMBL29929480 0.69 FLT3 (0.55) AXLNPC1ALDH1A1MAPTRAB9A
SCHEMBL15824969 0.69 HRH4 (0.46) PLAUF12NCF1NOS3NOS1
SCHEMBL29928610 0.69 MEN1 (0.49) AXLNCF1BACE1HRH4ALDH1A1
SCHEMBL5202901 0.68 COMT (0.58) PLAUF12NCF1NOS3NOS1
SCHEMBL8942018 0.67 TSHR (0.58) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL4635351 0.67 HRH4 (0.55) AXLPLAUF12NCF1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110551105-B Substituted triazoles useful as AXL inhibitors 里格尔制药公司 2022-10-18 CN claimed
CN-110551105-B Substituted triazoles useful as AXL inhibitors 里格尔制药公司 2022-10-18 CN disclosed